佩普医药始终瞄准新药发展的动向,以临床需求为导向,通过高效率设计、合成以及药理筛选,寻找结构新药的候选化合物,目前多个靶点的化合物已进入成药性研究阶段。
项目名称 | 疾病 | 靶点 | 研发阶段 | 备注 |
专注于小分子药物发现领域的分子砌块和工具化合物的研究开发,以及小分子药物原料药、中间体的工艺开发和生产技术改进。
CAS号 | 货号 | 产品名称 | 结构式 | |
1780780-13-3 | ||||
69008-41-9 | ||||
6683-46-1 | ||||
110952-37-9 | ||||
1883496-85-2 | ||||
2071683-27-5 | ||||
2007909-60-4 | ||||
903895-80-7 | ||||
2166023-31-8 | ||||
1374828-69-9 | ||||
1693734-80-3 | ||||
2275774-60-0 | ||||
2446480-97-1 | ||||
2411748-50-8 | ||||
1358751-06-0 | ||||
293762-45-5 | ||||
345952-44-5 | ||||
2756818-39-8 | ||||
2460249-19-6 | ||||
2762617-31-0 | ||||
2085274-00-4 | ||||
2376146-48-2 | ||||
2691879-68-0 | ||||
2691879-67-9 | ||||
2691869-82-4 | ||||
164341-39-3 | ||||
2719793-90-3 | ||||
2691878-21-2 | ||||
2589531-76-8 | ||||
1211538-09-8 | ||||
227321-68-8 | ||||
135748-35-5 | ||||
508203-26-7 | ||||
130255-28-6 | ||||
92775-34-3 | ||||
1936364-68-9 | ||||
885518-76-3 | ||||
143918-70-1 | ||||
205240-63-7 | ||||
2185857-89-8 | ||||
2185860-75-5 | ||||
2185860-74-4 | ||||
2185860-16-4 | ||||
2185860-12-0 | ||||
1354951-89-5 | ||||
2768088-21-5 | ||||
2768088-19-1 | ||||
908111-35-3 | ||||
908111-34-2 | ||||
2071683-99-1 | ||||
2757405-31-3 | ||||
2761063-99-2 | ||||
457657-34-0 | ||||
1845777-61-8 | ||||
2388506-43-0 | ||||
2388506-44-1 | ||||
1400689-45-3 | ||||
2185860-14-2 | ||||
118802-40-7 | ||||
1005333-24-3 | ||||
152754-30-8 | ||||
130255-27-5 | ||||
65818-01-1 | ||||
1628042-58-9 | ||||
338739-89-2 | ||||
15286-98-3 | ||||
5750-74-3 | ||||
1503948-15-9 | ||||
22190-35-8 | ||||
103796-41-4 | ||||
796854-35-8 | ||||
796856-20-7 | ||||
2100258-95-3 | ||||
2100258-94-2 | ||||
796853-76-4 | ||||
1246894-21-2 | ||||
7498-85-3 | ||||
454228-69-4 | ||||
2070931-57-4 | ||||
2070932-03-3 | ||||
2033057-23-5 | ||||
2033057-21-3 | ||||
2033057-22-4 | ||||
76872-68-9 | ||||
1029413-55-5 | ||||
35265-82-8 | ||||
35265-80-6 | ||||
5422-71-9 | ||||
6286-08-4 | ||||
2101843-64-3 | ||||
1845778-37-1 | ||||
2101830-25-3 | ||||
34121-17-0 | ||||
3086-91-7 | ||||
17560-53-1 | ||||
903895-98-7 | ||||
36193-65-4 | ||||
1670-84-4 | ||||
1698477-92-7 | ||||
856970-31-5 | ||||
1360883-22-2 | ||||
1863952-15-1 | ||||
2033057-23-5 | ||||
2033057-22-4 | ||||
2033057-21-3 | ||||
1201916-87-1 | ||||
35265-82-8 | ||||
2070931-57-4 | ||||
20287-37-0 | ||||
113293-70-2 | ||||
2244992-39-8 | ||||
1002309-52-5 | ||||
2245824-02-4 | ||||
2244987-03-7 | ||||
90182-92-6 | ||||
101303-98-4 | ||||
2185857-97-8 | ||||
1227593-77-2 | ||||
1227502-89-7 | ||||
2719749-02-5 | ||||
7169-93-9 | ||||
31052-95-6 | ||||
31040-18-3 | ||||
7169-91-7 | ||||
2229711-68-4 | ||||
3459-20-9 | ||||
339-44-6 | ||||
1945948-65-1 | ||||
3603-07-4 | ||||
2166027-04-7 | ||||
2166027-40-1 | ||||
2166027-03-6 | ||||
372198-41-9 | ||||
6052-73-9 | ||||
2757405-72-2 | ||||
2757405-73-3 | ||||
213211-10-0 | ||||
213208-73-2 | ||||
302840-67-1 | ||||
648422-58-6 | ||||
321724-17-8 | ||||
648422-57-5 | ||||
302840-64-8 | ||||
1698477-92-7 | PP2204032 | |||
856970-31-5 | PP2204031 | |||
1360883-22-2 | PP2204030 | |||
1863952-15-1 | PP2204029 | |||
2033057-23-5 | PP2204028 | |||
2033057-22-4 | PP2204027 | |||
2033057-21-3 | PP2204026 | |||
1201916-87-1 | PP2204025 | |||
35265-82-8 | PP2204024 | |||
2070931-57-4 | PP2204023 | |||
20287-37-0 | PP2204022 | |||
2304654-48-4 | PP2204021 | |||
1390656-66-2 | PP2204020 | |||
113293-70-2 | PP2204019 | |||
2304654-43-9 | PP2204018 | |||
2244992-39-8 | PP2204017 | |||
1002309-52-5 | PP2204016 | |||
2244987-03-7 | PP2204015 | |||
2245824-02-4 | PP2204014 | |||
90182-92-6 | PP2204013 | |||
101303-98-4 | PP2204012 | |||
2185857-97-8 | PP2204011 | |||
2629316-13-6 | PP2204010 | |||
2629316-03-4 | PP2204009 | |||
2629316-07-8 | PP2204008 | |||
2629316-02-3 | PP2204007 | |||
2629317-93-5 | PP2204006 | |||
2629317-94-6 | PP2204005 | |||
2629317-96-8 | PP2204004 | |||
2629317-95-7 | PP2204003 | |||
2629316-13-6 | PP2204002 | |||
2630904-45-7 | PP2204001 | |||
1227593-77-2 | PP2202007 | |||
1227502-89-7 | PP2202006 | |||
2719749-02-5 | PP2202005 | |||
7169-93-9 | PP2202004 | |||
31052-95-6 | PP2202003 | |||
31040-18-3 | PP2202002 | |||
7169-91-7 | PP2202001 | |||
61533-68-4 | PP2201054 | Glymidine | ||
1206117-96-5 | PP2201053 | |||
607-19-2 | PP2201052 | 5-(2-Methoxyethoxy)-2-pyrimidinamine | ||
138163-07-2 | PP2201051 | 2-chloro-5-(2-methoxyethoxy)pyrimidine | ||
29883-25-8 | PP2201050 | 3-methyl-2,4-dioxo-1,2,3,4-tetrahydro-6-quinazolinesulfonyl chloride | ||
151367-92-9 | PP2201049 | 3-Methylquinazoline-2,4(1H,3H)-dione | ||
2242744-56-3 | PP2201048 | (S)-3-Amino-piperidine-2,6-dione | ||
2741696-03-5 | PP2201047 | (S)-3-Boc-amino-2,6-dioxopiperidine | ||
2229713-89-5 | PP2201046 | |||
2229713-87-3 | PP2201045 | |||
2229713-85-1 | PP2201044 | |||
2229713-83-9 | PP2201043 | |||
2102527-98-8 | PP2201042 | |||
1273651-64-1 | PP2201041 | |||
1430472-11-9 | PP2201040 | |||
2129163-31-9 | PP2201039 | 6-(tert-Butoxy)-3,4-Dihydronaphthalen-1(2H)-one | ||
1639892-90-2 | PP2201038 | |||
372198-41-9 | PP2201037 | |||
2548-29-0 | PP2201036 | Methyl3-(chlorosulfonyl)-4-methylbenzoate | ||
2589531-73-5 | PP2201035 | 3-chlorosulfonyl-4-methyl-benzoic acid | ||
2589534-23-4 | PP2201034 | ethyl 7-Ethyl-6-oxo-5,6-dihydro-1,5-naphthyridine-3-carboxylate | ||
2589531-70-2 | PP2201033 | |||
2589534-19-8 | PP2201032 | |||
1354355-85-3 | PP2201031 | |||
1211538-09-8 | PP2201030 | tert-Butyl 4-(6-(methoxycarbonyl)pyridin-3-yl)piperazine-1-carboxylate | ||
2382997-02-4 | PP2201029 | ethyl 6-methyl-5-nitropyridine-3-carboxylate | ||
95645-00-4 | PP2201028 | |||
81115-59-5 | PP2201027 | 3-methoxy-2,6-dimethylaniline | ||
95644-98-7 | PP2201026 | 5-methyl-4-nitro-1H-indazole | ||
53874-26-3 | PP2201025 | |||
31167-04-1 | PP2201024 | 3-BroMo-2,6-diMetylaniline | ||
39053-43-5 | PP2201023 | 1-Bromo-2,4-dimethyl-3-nitro-benzene | ||
18520-07-5 | PP2201022 | |||
62409-52-3 | PP2201021 | 2,6-Dichloro-4-ethyl-3,5-pyridinedicarbonitrile | ||
2422150-99-8 | PP2201020 | (5S)-5-Phenylmorpholin-2-one Hydrochloride | ||
2170142-58-0 | PP2201019 | Ethyl2-chloro-5-fluoropyridine-3-carboxylate | ||
2170140-50-6 | PP2201018 | |||
2170137-61-6 | PP2201017 | |||
2520107-65-5 | PP2201016 | |||
2097342-14-6 | PP2201015 | NCGC00029283 | ||
2201057-82-9 | PP2201014 | |||
2201057-80-7 | PP2201013 | 4-(Cyclohex-1-en-1-yl)-3-phenyl-1h-pyrazol-5-amine | ||
2201057-79-4 | PP2201012 | |||
2201058-77-5 | PP2201011 | |||
2201058-76-4 | PP2201010 | |||
899937-47-4 | PP2201009 | 3-[(METHYLSULFONYL)METHYL]BENZENAMINE | ||
1370885-46-3 | PP2201008 | |||
2197052-44-9 | PP2201007 | 4-Hydroxyquinoline-3-carboxaldehyde | ||
2381044-63-7 | PP2201006 | NA | ||
745066-18-6 | PP2201005 | |||
2381043-66-7 | PP2201004 | 2-(哌嗪-1-基)-5-三氟甲基嘧啶 | ||
1599440-07-9 | PP2201003 | |||
1330785-12-0 | PP2201002 | |||
2408929-29-1 | PP2201001 | |||
104421-21-8 | PP2110034 | Dup-721 | ||
1330782-76-7 | PP2110033 | TAK-931 | ||
52601-23-7 | PP2110030 | quinuiclidine-2-carboxylic acid hydrochloride | ||
714240-31-0 | PP2110028 | NCGC00029283 | ||
123990-79-4 | PP2110027 | 6-methoxy-2-oxo-1,2-dihydroquinoline-3-carbonitrile | ||
2201056-66-6 | PP2110026 | AG-270 | ||
261925-02-4 | PP2110017 | 3-((methylsulfonyl)methyl)aniline | ||
1042433-41-9 | PP2110016 | GSK-1520489A | ||
1022964-14-2 | PP2110015 | 2-[(2-chloro-5-methylpyrimidin-4-yl)amino]-N-methylbenzamide | ||
261924-46-3 | PP2110014 | 1-(methylsulfonylmethyl)-3-nitrobenzene | ||
82121-18-4或者83342-32-9 | PP2110012 | 4-hydroxy-3-hydroxymethylquinoline | ||
7509-12-8或者83342-70-5 | PP2110011 | 1,4-dihydro-4-oxoquinoline-3-carbaldehyde | ||
71879-53-3 | PP2110003 | diethyl (piperidin-4-ylmethyl)propanedioate | ||
13738-70-0 | PP2110001 | 4-[(Phenylsulfanyl)methyl]aniline | ||
1352707-53-9 | PP2105035 | 1',3'-propanedisulfonyl (L)-rhamnose | ||
491833-30-8 | PP2105034 | Genz-123346 | ||
491833-29-5 | PP2105033 | Eliglustat | ||
14464-30-3 | PP2105032 | N-succinimidyl caprylate | ||
491833-27-3 | PP2105031 | (1R,2R)-1-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-2-((2-hydroxy-1-phenylethyl)amino)-3-(pyrrolidin-1-yl)propan-1-ol | ||
491833-26-2 | PP2105030 | (2S,3R)-3-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-3-hydroxy-2-((2-hydroxy-1-phenylethyl)amino)-1-(pyrrolidin-1-yl)propan-1-one | ||
29668-44-8 | PP2105029 | 1,4-Benzodioxan-6-carboxaldehyde | ||
491833-36-4 | PP2105028 | (5S)-5-Phenyl-2-morpholinone hydrochloride | ||
1306760-87-1 | PP2105027 | Ozanimod | ||
82304-99-2 | PP2105026 | ethyl 3-formyl-4-hydroxybenzoate | ||
258273-31-3 | PP2105025 | 3-Cyano-4-isopropoxy-benzoic acid methyl ester | ||
1306763-61-0 | PP2105024 | (S)-tert-butyl (2-((tert-butyldimethylsilyl)oxy)ethyl)(4-cyano-2,3-dihydro-1H-inden-1-yl)carbamate | ||
1306763-31-4 | PP2105023 | (R)-tert-butyl (4-cyano-2,3-dihydro-1H-inden-1-yl)carbamate | ||
1306763-57-4 | PP2105022 | (S)-1-amino-2,3-dihydro-1H-indene-4-carbonitrile hydrochloride | ||
60899-34-5 | PP2105021 | 2,3-dihydro-1-oxo-1H-indene-4-carbonitrile | ||
249921-19-5 | PP2105020 | Anamorelin | ||
339539-90-1 | PP2105019 | tert-butyl (1-(((R)-1-((R)-3-benzyl-3-(1,2,2-trimethylhydrazine-1-carbonyl)piperidin-1-yl)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)amino)-2-methyl-1-oxopropan-2-yl)carbamate | ||
159634-94-3 | PP2105018 | (R)-2-(2-((tert-Butoxycarbonyl)amino)-2-methylpropanamido)-3-(1H-indol-3-yl)propanoic acid | ||
185056-99-9 | PP2105017 | methyl (2-((tert-butoxycarbonyl)amino)-2-methylpropanoyl)-D-tryptophanate | ||
339539-84-3 | PP2105016 | (3R)-3-Benzyl-piperidine-3-carboxylic acid triMethylhydrazide hydrochloride | ||
339539-82-1 | PP2105015 | tert-butyl (R)-3-benzyl-3-(1,2,2-trimethylhydrazine-1-carbonyl)piperidine-1-carboxylate | ||
339539-81-0 | PP2105014 | (R)-3-benzyl-1-(tert-butoxycarbonyl)piperidine-3-carboxylic acid | ||
170838-83-2 | PP2105013 | 3-Benzyl-piperidine-1,3-dicarboxylic acid 1-tert-butyl ester | ||
170842-80-5 | PP2105012 | Ethyl 1-Boc-3-benzylpiperidine-3-carboxylate | ||
824932-88-9 | PP2105011 | Elafibranor | ||
1000335-03-4 | PP2105010 | isopropyl (E)-2-(2,6-dimethyl-4-(3-(4-(methylthio)phenyl)-3-oxoprop-1-en-1-yl)phenoxy)-2-methylpropanoate | ||
824932-89-0 | PP2105009 | 1-[4-methylthiophenyl]-3-[3,5-dimethyl-4-hydroxyphenyl]prop-2-en-1-one | ||
2097002-61-2 | PP2105008 | LOXO-195 | ||
/ | PP2105007 | ethyl 5-((R)-2-(2-((R)-3-((tert-butoxycarbonyl)amino)butyl)-5-fluoropyridin-3-yl)pyrrolidin-1-yl)pyrazolo[1,5-a]pyrimidine-3-carboxylate | ||
1224944-77-7 | PP2105006 | Ethyl 5-chloropyrazolo[1,5-a]pyrimidine-3-carboxylate | ||
167216-17-3 | PP2105005 | N-Boc-(R)-3-aminobutan-1-ol | ||
1260847-45-7 | PP2105004 | (R)-2-chloro-5-fluoro-3-(pyrrolidin-2-yl)pyridine dihydrochloride | ||
851484-95-2 | PP2105003 | 2-Chloro-5-fluoropyridine-3-carbaldehyde | ||
847729-27-5 | PP2105002 | Methyl 2-chloro-5-fluoronicotinate | ||
139911-30-1 | PP2105001 | ethyl 2-chloro-5-fluoronicotinate |