创新药研发管线

佩普医药始终瞄准新药发展的动向,以临床需求为导向,通过高效率设计、合成以及药理筛选,寻找结构新药的候选化合物,目前多个靶点的化合物已进入成药性研究阶段。


项目名称 疾病 靶点 研发阶段 备注
药物及中间体

专注于小分子药物发现领域的分子砌块和工具化合物的研究开发,以及小分子药物原料药、中间体的工艺开发和生产技术改进。


CAS号 货号 产品名称 结构式
1780780-13-3

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69008-41-9

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6683-46-1

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110952-37-9

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1883496-85-2

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2071683-27-5

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2007909-60-4

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903895-80-7

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2166023-31-8

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1374828-69-9

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1693734-80-3

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2275774-60-0

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2446480-97-1

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2411748-50-8

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1358751-06-0

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293762-45-5

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345952-44-5

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2756818-39-8

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2460249-19-6

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2762617-31-0

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2085274-00-4

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2376146-48-2

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2691879-68-0

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2691879-67-9

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2691869-82-4

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164341-39-3

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2719793-90-3

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2691878-21-2

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2589531-76-8

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1211538-09-8

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227321-68-8

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135748-35-5

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508203-26-7

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130255-28-6

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92775-34-3

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1936364-68-9

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885518-76-3

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143918-70-1

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205240-63-7

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2185857-89-8

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2185860-75-5

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2185860-74-4

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2185860-16-4

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2185860-12-0

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1354951-89-5

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2768088-21-5

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2768088-19-1

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908111-35-3

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908111-34-2

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2071683-99-1

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2757405-31-3

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2761063-99-2

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457657-34-0

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1845777-61-8

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2388506-43-0

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2388506-44-1

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1400689-45-3

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2185860-14-2

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118802-40-7

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1005333-24-3

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152754-30-8

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130255-27-5

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65818-01-1

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1628042-58-9

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338739-89-2

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15286-98-3

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5750-74-3

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1503948-15-9

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22190-35-8

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103796-41-4

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796854-35-8

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796856-20-7

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2100258-95-3

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2100258-94-2

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796853-76-4

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1246894-21-2

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7498-85-3

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454228-69-4

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2070931-57-4

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2070932-03-3

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2033057-23-5

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2033057-21-3

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2033057-22-4

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76872-68-9

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1029413-55-5

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35265-82-8

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35265-80-6

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5422-71-9

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6286-08-4

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2101843-64-3

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1845778-37-1

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2101830-25-3

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34121-17-0

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3086-91-7

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17560-53-1

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903895-98-7

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36193-65-4

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1670-84-4

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1698477-92-7

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856970-31-5

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1360883-22-2

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1863952-15-1

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2033057-23-5

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2033057-22-4

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2033057-21-3

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1201916-87-1

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35265-82-8

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2070931-57-4

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20287-37-0

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113293-70-2

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2244992-39-8

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1002309-52-5

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2245824-02-4

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2244987-03-7

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90182-92-6

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101303-98-4

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2185857-97-8

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1227593-77-2

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1227502-89-7

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2719749-02-5

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7169-93-9

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31052-95-6


31040-18-3

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7169-91-7

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2229711-68-4

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3459-20-9

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339-44-6

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1945948-65-1

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3603-07-4

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2166027-04-7

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2166027-40-1

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2166027-03-6

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372198-41-9

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6052-73-9

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2757405-72-2

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2757405-73-3

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213211-10-0

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213208-73-2

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302840-67-1

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648422-58-6

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321724-17-8

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648422-57-5

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302840-64-8

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1698477-92-7 PP2204032

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856970-31-5 PP2204031

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1360883-22-2 PP2204030

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1863952-15-1 PP2204029

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2033057-23-5 PP2204028

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2033057-22-4 PP2204027

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2033057-21-3 PP2204026

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 1201916-87-1 PP2204025

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35265-82-8 PP2204024

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2070931-57-4 PP2204023

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20287-37-0 PP2204022

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2304654-48-4 PP2204021

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1390656-66-2 PP2204020

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113293-70-2 PP2204019

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2304654-43-9 PP2204018

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2244992-39-8 PP2204017

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1002309-52-5 PP2204016

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2244987-03-7 PP2204015

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 2245824-02-4 PP2204014

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90182-92-6 PP2204013

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101303-98-4 PP2204012

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2185857-97-8 PP2204011

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2629316-13-6 PP2204010

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2629316-03-4 PP2204009

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2629316-07-8 PP2204008

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2629316-02-3 PP2204007

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2629317-93-5 PP2204006

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2629317-94-6 PP2204005

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2629317-96-8 PP2204004

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2629317-95-7 PP2204003

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 2629316-13-6 PP2204002

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2630904-45-7 PP2204001

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1227593-77-2 PP2202007

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1227502-89-7 PP2202006

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2719749-02-5 PP2202005

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7169-93-9 PP2202004

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31052-95-6 PP2202003

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31040-18-3 PP2202002

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7169-91-7 PP2202001

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61533-68-4 PP2201054 Glymidine

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1206117-96-5 PP2201053

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607-19-2 PP2201052 5-(2-Methoxyethoxy)-2-pyrimidinamine

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138163-07-2 PP2201051 2-chloro-5-(2-methoxyethoxy)pyrimidine

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29883-25-8 PP2201050 3-methyl-2,4-dioxo-1,2,3,4-tetrahydro-6-quinazolinesulfonyl chloride

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151367-92-9 PP2201049 3-Methylquinazoline-2,4(1H,3H)-dione

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2242744-56-3 PP2201048 (S)-3-Amino-piperidine-2,6-dione

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2741696-03-5 PP2201047 (S)-3-Boc-amino-2,6-dioxopiperidine

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2229713-89-5 PP2201046

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2229713-87-3 PP2201045

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2229713-85-1 PP2201044

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2229713-83-9 PP2201043

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2102527-98-8 PP2201042

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1273651-64-1 PP2201041

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1430472-11-9 PP2201040

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2129163-31-9 PP2201039 6-(tert-Butoxy)-3,4-Dihydronaphthalen-1(2H)-one

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1639892-90-2 PP2201038

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372198-41-9 PP2201037

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2548-29-0 PP2201036 Methyl3-(chlorosulfonyl)-4-methylbenzoate

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2589531-73-5 PP2201035 3-chlorosulfonyl-4-methyl-benzoic acid

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2589534-23-4 PP2201034 ethyl 7-Ethyl-6-oxo-5,6-dihydro-1,5-naphthyridine-3-carboxylate

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2589531-70-2 PP2201033

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2589534-19-8 PP2201032

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1354355-85-3 PP2201031

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1211538-09-8 PP2201030 tert-Butyl 4-(6-(methoxycarbonyl)pyridin-3-yl)piperazine-1-carboxylate

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2382997-02-4 PP2201029 ethyl 6-methyl-5-nitropyridine-3-carboxylate

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95645-00-4 PP2201028

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81115-59-5 PP2201027 3-methoxy-2,6-dimethylaniline

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95644-98-7 PP2201026 5-methyl-4-nitro-1H-indazole

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53874-26-3 PP2201025

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31167-04-1 PP2201024 3-BroMo-2,6-diMetylaniline

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39053-43-5 PP2201023 1-Bromo-2,4-dimethyl-3-nitro-benzene

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18520-07-5 PP2201022

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62409-52-3 PP2201021 2,6-Dichloro-4-ethyl-3,5-pyridinedicarbonitrile

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2422150-99-8 PP2201020 (5S)-5-Phenylmorpholin-2-one Hydrochloride

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2170142-58-0 PP2201019 Ethyl2-chloro-5-fluoropyridine-3-carboxylate

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2170140-50-6 PP2201018

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2170137-61-6 PP2201017

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2520107-65-5 PP2201016

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2097342-14-6 PP2201015 NCGC00029283

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2201057-82-9 PP2201014

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2201057-80-7 PP2201013 4-(Cyclohex-1-en-1-yl)-3-phenyl-1h-pyrazol-5-amine

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2201057-79-4 PP2201012

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2201058-77-5 PP2201011

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2201058-76-4 PP2201010

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899937-47-4 PP2201009 3-[(METHYLSULFONYL)METHYL]BENZENAMINE

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1370885-46-3 PP2201008

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2197052-44-9 PP2201007 4-Hydroxyquinoline-3-carboxaldehyde

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2381044-63-7 PP2201006 NA

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745066-18-6 PP2201005

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2381043-66-7 PP2201004 2-(哌嗪-1-基)-5-三氟甲基嘧啶

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1599440-07-9 PP2201003

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1330785-12-0 PP2201002

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2408929-29-1 PP2201001

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104421-21-8 PP2110034 Dup-721

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1330782-76-7 PP2110033 TAK-931

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52601-23-7 PP2110030 quinuiclidine-2-carboxylic acid hydrochloride

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714240-31-0 PP2110028 NCGC00029283

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123990-79-4 PP2110027 6-methoxy-2-oxo-1,2-dihydroquinoline-3-carbonitrile

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2201056-66-6 PP2110026 AG-270

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261925-02-4 PP2110017 3-((methylsulfonyl)methyl)aniline

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1042433-41-9 PP2110016 GSK-1520489A

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1022964-14-2 PP2110015 2-[(2-chloro-5-methylpyrimidin-4-yl)amino]-N-methylbenzamide

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261924-46-3 PP2110014 1-(methylsulfonylmethyl)-3-nitrobenzene

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82121-18-4或者83342-32-9 PP2110012 4-hydroxy-3-hydroxymethylquinoline

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7509-12-8或者83342-70-5 PP2110011 1,4-dihydro-4-oxoquinoline-3-carbaldehyde

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71879-53-3 PP2110003 diethyl (piperidin-4-ylmethyl)propanedioate

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13738-70-0 PP2110001 4-[(Phenylsulfanyl)methyl]aniline

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1352707-53-9 PP2105035 1',3'-propanedisulfonyl (L)-rhamnose

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491833-30-8 PP2105034 Genz-123346

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491833-29-5 PP2105033 Eliglustat

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14464-30-3 PP2105032 N-succinimidyl caprylate

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491833-27-3 PP2105031 (1R,2R)-1-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-2-((2-hydroxy-1-phenylethyl)amino)-3-(pyrrolidin-1-yl)propan-1-ol

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491833-26-2 PP2105030 (2S,3R)-3-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-3-hydroxy-2-((2-hydroxy-1-phenylethyl)amino)-1-(pyrrolidin-1-yl)propan-1-one

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29668-44-8 PP2105029 1,4-Benzodioxan-6-carboxaldehyde

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491833-36-4 PP2105028 (5S)-5-Phenyl-2-morpholinone hydrochloride

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1306760-87-1 PP2105027 Ozanimod

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82304-99-2 PP2105026 ethyl 3-formyl-4-hydroxybenzoate

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258273-31-3 PP2105025 3-Cyano-4-isopropoxy-benzoic acid methyl ester

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1306763-61-0 PP2105024 (S)-tert-butyl (2-((tert-butyldimethylsilyl)oxy)ethyl)(4-cyano-2,3-dihydro-1H-inden-1-yl)carbamate

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1306763-31-4 PP2105023 (R)-tert-butyl (4-cyano-2,3-dihydro-1H-inden-1-yl)carbamate

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1306763-57-4 PP2105022 (S)-1-amino-2,3-dihydro-1H-indene-4-carbonitrile hydrochloride

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60899-34-5 PP2105021 2,3-dihydro-1-oxo-1H-indene-4-carbonitrile

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249921-19-5 PP2105020 Anamorelin

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339539-90-1 PP2105019 tert-butyl (1-(((R)-1-((R)-3-benzyl-3-(1,2,2-trimethylhydrazine-1-carbonyl)piperidin-1-yl)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)amino)-2-methyl-1-oxopropan-2-yl)carbamate

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159634-94-3 PP2105018 (R)-2-(2-((tert-Butoxycarbonyl)amino)-2-methylpropanamido)-3-(1H-indol-3-yl)propanoic acid

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185056-99-9 PP2105017 methyl (2-((tert-butoxycarbonyl)amino)-2-methylpropanoyl)-D-tryptophanate

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339539-84-3 PP2105016 (3R)-3-Benzyl-piperidine-3-carboxylic acid triMethylhydrazide hydrochloride

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339539-82-1 PP2105015 tert-butyl (R)-3-benzyl-3-(1,2,2-trimethylhydrazine-1-carbonyl)piperidine-1-carboxylate

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339539-81-0 PP2105014 (R)-3-benzyl-1-(tert-butoxycarbonyl)piperidine-3-carboxylic acid

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170838-83-2 PP2105013 3-Benzyl-piperidine-1,3-dicarboxylic acid 1-tert-butyl ester

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170842-80-5 PP2105012 Ethyl 1-Boc-3-benzylpiperidine-3-carboxylate

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824932-88-9 PP2105011 Elafibranor

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1000335-03-4 PP2105010 isopropyl (E)-2-(2,6-dimethyl-4-(3-(4-(methylthio)phenyl)-3-oxoprop-1-en-1-yl)phenoxy)-2-methylpropanoate

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824932-89-0 PP2105009 1-[4-methylthiophenyl]-3-[3,5-dimethyl-4-hydroxyphenyl]prop-2-en-1-one

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2097002-61-2 PP2105008 LOXO-195

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/ PP2105007 ethyl 5-((R)-2-(2-((R)-3-((tert-butoxycarbonyl)amino)butyl)-5-fluoropyridin-3-yl)pyrrolidin-1-yl)pyrazolo[1,5-a]pyrimidine-3-carboxylate

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1224944-77-7 PP2105006 Ethyl 5-chloropyrazolo[1,5-a]pyrimidine-3-carboxylate

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167216-17-3 PP2105005 N-Boc-(R)-3-aminobutan-1-ol

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1260847-45-7 PP2105004 (R)-2-chloro-5-fluoro-3-(pyrrolidin-2-yl)pyridine dihydrochloride

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851484-95-2 PP2105003 2-Chloro-5-fluoropyridine-3-carbaldehyde

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847729-27-5 PP2105002 Methyl 2-chloro-5-fluoronicotinate

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139911-30-1 PP2105001 ethyl 2-chloro-5-fluoronicotinate

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