佩普医药始终瞄准新药发展的动向,以临床需求为导向,通过高效率设计、合成以及药理筛选,寻找结构新药的候选化合物,目前多个靶点的化合物已进入成药性研究阶段。
项目名称 | 疾病 | 靶点 | 研发阶段 | 备注 |
专注于小分子药物发现领域的分子砌块和工具化合物的研究开发,以及小分子药物原料药、中间体的工艺开发和生产技术改进。
CAS号 | 货号 | 产品名称 | 结构式 |
1698477-92-7 | PP2204032 | ||
856970-31-5 | PP2204031 | ||
1360883-22-2 | PP2204030 | ||
1863952-15-1 | PP2204029 | ||
2033057-23-5 | PP2204028 | ||
2033057-22-4 | PP2204027 | ||
2033057-21-3 | PP2204026 | ||
1201916-87-1 | PP2204025 | ||
35265-82-8 | PP2204024 | ||
2070931-57-4 | PP2204023 | ||
20287-37-0 | PP2204022 | ||
2304654-48-4 | PP2204021 | ||
1390656-66-2 | PP2204020 | ||
113293-70-2 | PP2204019 | ||
2304654-43-9 | PP2204018 | ||
2244992-39-8 | PP2204017 | ||
1002309-52-5 | PP2204016 | ||
2244987-03-7 | PP2204015 | ||
2245824-02-4 | PP2204014 | ||
90182-92-6 | PP2204013 | ||
101303-98-4 | PP2204012 | ||
2185857-97-8 | PP2204011 | ||
2629316-13-6 | PP2204010 | ||
2629316-03-4 | PP2204009 | ||
2629316-07-8 | PP2204008 | ||
2629316-02-3 | PP2204007 | ||
2629317-93-5 | PP2204006 | ||
2629317-94-6 | PP2204005 | ||
2629317-96-8 | PP2204004 | ||
2629317-95-7 | PP2204003 | ||
2629316-13-6 | PP2204002 | ||
2630904-45-7 | PP2204001 | ||
1227593-77-2 | PP2202007 | ||
1227502-89-7 | PP2202006 | ||
2719749-02-5 | PP2202005 | ||
7169-93-9 | PP2202004 | ||
31052-95-6 | PP2202003 | ||
31040-18-3 | PP2202002 | ||
7169-91-7 | PP2202001 | ||
61533-68-4 | PP2201054 | Glymidine | |
1206117-96-5 | PP2201053 | ||
607-19-2 | PP2201052 | 5-(2-Methoxyethoxy)-2-pyrimidinamine | |
138163-07-2 | PP2201051 | 2-chloro-5-(2-methoxyethoxy)pyrimidine | |
29883-25-8 | PP2201050 | 3-methyl-2,4-dioxo-1,2,3,4-tetrahydro-6-quinazolinesulfonyl chloride | |
151367-92-9 | PP2201049 | 3-Methylquinazoline-2,4(1H,3H)-dione | |
2242744-56-3 | PP2201048 | (S)-3-Amino-piperidine-2,6-dione | |
2741696-03-5 | PP2201047 | (S)-3-Boc-amino-2,6-dioxopiperidine | |
2229713-89-5 | PP2201046 | ||
2229713-87-3 | PP2201045 | ||
2229713-85-1 | PP2201044 | ||
2229713-83-9 | PP2201043 | ||
2102527-98-8 | PP2201042 | ||
1273651-64-1 | PP2201041 | ||
1430472-11-9 | PP2201040 | ||
2129163-31-9 | PP2201039 | 6-(tert-Butoxy)-3,4-Dihydronaphthalen-1(2H)-one | |
1639892-90-2 | PP2201038 | ||
372198-41-9 | PP2201037 | ||
2548-29-0 | PP2201036 | Methyl3-(chlorosulfonyl)-4-methylbenzoate | |
2589531-73-5 | PP2201035 | 3-chlorosulfonyl-4-methyl-benzoic acid | |
2589534-23-4 | PP2201034 | ethyl 7-Ethyl-6-oxo-5,6-dihydro-1,5-naphthyridine-3-carboxylate | |
2589531-70-2 | PP2201033 | ||
2589534-19-8 | PP2201032 | ||
1354355-85-3 | PP2201031 | ||
1211538-09-8 | PP2201030 | tert-Butyl 4-(6-(methoxycarbonyl)pyridin-3-yl)piperazine-1-carboxylate | |
2382997-02-4 | PP2201029 | ethyl 6-methyl-5-nitropyridine-3-carboxylate | |
95645-00-4 | PP2201028 | ||
81115-59-5 | PP2201027 | 3-methoxy-2,6-dimethylaniline | |
95644-98-7 | PP2201026 | 5-methyl-4-nitro-1H-indazole | |
53874-26-3 | PP2201025 | ||
31167-04-1 | PP2201024 | 3-BroMo-2,6-diMetylaniline | |
39053-43-5 | PP2201023 | 1-Bromo-2,4-dimethyl-3-nitro-benzene | |
18520-07-5 | PP2201022 | ||
62409-52-3 | PP2201021 | 2,6-Dichloro-4-ethyl-3,5-pyridinedicarbonitrile | |
2422150-99-8 | PP2201020 | (5S)-5-Phenylmorpholin-2-one Hydrochloride | |
2170142-58-0 | PP2201019 | Ethyl2-chloro-5-fluoropyridine-3-carboxylate | |
2170140-50-6 | PP2201018 | ||
2170137-61-6 | PP2201017 | ||
2520107-65-5 | PP2201016 | ||
2097342-14-6 | PP2201015 | NCGC00029283 | |
2201057-82-9 | PP2201014 | ||
2201057-80-7 | PP2201013 | 4-(Cyclohex-1-en-1-yl)-3-phenyl-1h-pyrazol-5-amine | |
2201057-79-4 | PP2201012 | ||
2201058-77-5 | PP2201011 | ||
2201058-76-4 | PP2201010 | ||
899937-47-4 | PP2201009 | 3-[(METHYLSULFONYL)METHYL]BENZENAMINE | |
1370885-46-3 | PP2201008 | ||
2197052-44-9 | PP2201007 | 4-Hydroxyquinoline-3-carboxaldehyde | |
2381044-63-7 | PP2201006 | NA | |
745066-18-6 | PP2201005 | ||
2381043-66-7 | PP2201004 | 2-(哌嗪-1-基)-5-三氟甲基嘧啶 | |
1599440-07-9 | PP2201003 | ||
1330785-12-0 | PP2201002 | ||
2408929-29-1 | PP2201001 | ||
104421-21-8 | PP2110034 | Dup-721 | |
1330782-76-7 | PP2110033 | TAK-931 | |
52601-23-7 | PP2110030 | quinuiclidine-2-carboxylic acid hydrochloride | |
714240-31-0 | PP2110028 | NCGC00029283 | |
123990-79-4 | PP2110027 | 6-methoxy-2-oxo-1,2-dihydroquinoline-3-carbonitrile | |
2201056-66-6 | PP2110026 | AG-270 | |
261925-02-4 | PP2110017 | 3-((methylsulfonyl)methyl)aniline | |
1042433-41-9 | PP2110016 | GSK-1520489A | |
1022964-14-2 | PP2110015 | 2-[(2-chloro-5-methylpyrimidin-4-yl)amino]-N-methylbenzamide | |
261924-46-3 | PP2110014 | 1-(methylsulfonylmethyl)-3-nitrobenzene | |
82121-18-4或者83342-32-9 | PP2110012 | 4-hydroxy-3-hydroxymethylquinoline | |
7509-12-8或者83342-70-5 | PP2110011 | 1,4-dihydro-4-oxoquinoline-3-carbaldehyde | |
71879-53-3 | PP2110003 | diethyl (piperidin-4-ylmethyl)propanedioate | |
13738-70-0 | PP2110001 | 4-[(Phenylsulfanyl)methyl]aniline | |
1352707-53-9 | PP2105035 | 1',3'-propanedisulfonyl (L)-rhamnose | |
491833-30-8 | PP2105034 | Genz-123346 | |
491833-29-5 | PP2105033 | Eliglustat | |
14464-30-3 | PP2105032 | N-succinimidyl caprylate | |
491833-27-3 | PP2105031 | (1R,2R)-1-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-2-((2-hydroxy-1-phenylethyl)amino)-3-(pyrrolidin-1-yl)propan-1-ol | |
491833-26-2 | PP2105030 | (2S,3R)-3-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-3-hydroxy-2-((2-hydroxy-1-phenylethyl)amino)-1-(pyrrolidin-1-yl)propan-1-one | |
29668-44-8 | PP2105029 | 1,4-Benzodioxan-6-carboxaldehyde | |
491833-36-4 | PP2105028 | (5S)-5-Phenyl-2-morpholinone hydrochloride | |
1306760-87-1 | PP2105027 | Ozanimod | |
82304-99-2 | PP2105026 | ethyl 3-formyl-4-hydroxybenzoate | |
258273-31-3 | PP2105025 | 3-Cyano-4-isopropoxy-benzoic acid methyl ester | |
1306763-61-0 | PP2105024 | (S)-tert-butyl (2-((tert-butyldimethylsilyl)oxy)ethyl)(4-cyano-2,3-dihydro-1H-inden-1-yl)carbamate | |
1306763-31-4 | PP2105023 | (R)-tert-butyl (4-cyano-2,3-dihydro-1H-inden-1-yl)carbamate | |
1306763-57-4 | PP2105022 | (S)-1-amino-2,3-dihydro-1H-indene-4-carbonitrile hydrochloride | |
60899-34-5 | PP2105021 | 2,3-dihydro-1-oxo-1H-indene-4-carbonitrile | |
249921-19-5 | PP2105020 | Anamorelin | |
339539-90-1 | PP2105019 | tert-butyl (1-(((R)-1-((R)-3-benzyl-3-(1,2,2-trimethylhydrazine-1-carbonyl)piperidin-1-yl)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)amino)-2-methyl-1-oxopropan-2-yl)carbamate | |
159634-94-3 | PP2105018 | (R)-2-(2-((tert-Butoxycarbonyl)amino)-2-methylpropanamido)-3-(1H-indol-3-yl)propanoic acid | |
185056-99-9 | PP2105017 | methyl (2-((tert-butoxycarbonyl)amino)-2-methylpropanoyl)-D-tryptophanate | |
339539-84-3 | PP2105016 | (3R)-3-Benzyl-piperidine-3-carboxylic acid triMethylhydrazide hydrochloride | |
339539-82-1 | PP2105015 | tert-butyl (R)-3-benzyl-3-(1,2,2-trimethylhydrazine-1-carbonyl)piperidine-1-carboxylate | |
339539-81-0 | PP2105014 | (R)-3-benzyl-1-(tert-butoxycarbonyl)piperidine-3-carboxylic acid | |
170838-83-2 | PP2105013 | 3-Benzyl-piperidine-1,3-dicarboxylic acid 1-tert-butyl ester | |
170842-80-5 | PP2105012 | Ethyl 1-Boc-3-benzylpiperidine-3-carboxylate | |
824932-88-9 | PP2105011 | Elafibranor | |
1000335-03-4 | PP2105010 | isopropyl (E)-2-(2,6-dimethyl-4-(3-(4-(methylthio)phenyl)-3-oxoprop-1-en-1-yl)phenoxy)-2-methylpropanoate | |
824932-89-0 | PP2105009 | 1-[4-methylthiophenyl]-3-[3,5-dimethyl-4-hydroxyphenyl]prop-2-en-1-one | |
2097002-61-2 | PP2105008 | LOXO-195 | |
/ | PP2105007 | ethyl 5-((R)-2-(2-((R)-3-((tert-butoxycarbonyl)amino)butyl)-5-fluoropyridin-3-yl)pyrrolidin-1-yl)pyrazolo[1,5-a]pyrimidine-3-carboxylate | |
1224944-77-7 | PP2105006 | Ethyl 5-chloropyrazolo[1,5-a]pyrimidine-3-carboxylate | |
167216-17-3 | PP2105005 | N-Boc-(R)-3-aminobutan-1-ol | |
1260847-45-7 | PP2105004 | (R)-2-chloro-5-fluoro-3-(pyrrolidin-2-yl)pyridine dihydrochloride | |
851484-95-2 | PP2105003 | 2-Chloro-5-fluoropyridine-3-carbaldehyde | |
847729-27-5 | PP2105002 | Methyl 2-chloro-5-fluoronicotinate | |
139911-30-1 | PP2105001 | ethyl 2-chloro-5-fluoronicotinate |